发明名称 N-cyanomethylamides as protease inhibitors.
摘要 The present invention relates to novel N-cyanomethyl amides which are cysteine protease inhibitors, the pharmaceutically acceptable salts and N-oxides thereof, their uses as therapeutic agents and the methods of their making.
申请公布号 ZA200107494(B) 申请公布日期 2002.11.27
申请号 ZA20010007494 申请日期 2001.09.11
申请人 AXYS PHARMACEUTICALS, INC. 发明人 CLIFFORD M BRYANT;JAMES T PALMER;ROBERT M RYDZEWSKI;EDUARDO L SETTI;ZONG-QIANG TIAN;SHANKAR VENKATRAMAN;DAN-XIONG WANG
分类号 C07D295/12;A61K31/275;A61K31/277;A61K31/341;A61K31/343;A61K31/36;A61K31/381;A61K31/395;A61K31/40;A61K31/404;A61K31/4045;A61K31/4164;A61K31/4166;A61K31/417;A61K31/426;A61K31/433;A61K31/4402;A61K31/4406;A61K31/4409;A61K31/4436;A61K31/4439;A61K31/445;A61K31/4453;A61K31/4468;A61K31/454;A61K31/455;A61K31/465;A61K31/47;A61K31/495;A61K31/496;A61K31/505;A61K31/535;A61K31/5375;A61K31/54;A61K31/663;A61K45/00;A61P3/10;A61P5/14;A61P9/00;A61P9/10;A61P11/00;A61P11/06;A61P17/00;A61P17/02;A61P19/02;A61P19/10;A61P21/04;A61P25/00;A61P25/28;A61P27/02;A61P29/00;A61P33/00;A61P35/00;A61P37/00;A61P37/02;A61P37/08;A61P43/00;C07C253/30;C07C255/29;C07C255/60;C07C269/06;C07C271/22;C07C273/18;C07C275/24;C07C303/40;C07C311/06;C07C311/09;C07C315/04;C07C317/50;C07C319/20;C07C323/52;C07C323/60;C07C323/62;C07D207/09;C07D207/14;C07D207/16;C07D209/06;C07D209/08;C07D209/14;C07D209/22;C07D209/26;C07D209/42;C07D209/52;C07D211/58;C07D211/60;C07D211/62;C07D213/30;C07D213/34;C07D213/40;C07D213/56;C07D213/70;C07D213/71;C07D213/75;C07D213/81;C07D213/82;C07D215/54;C07D233/24;C07D233/26;C07D233/64;C07D233/90;C07D239/28;C07D239/36;C07D277/20;C07D277/28;C07D277/30;C07D277/42;C07D277/48;C07D277/56;C07D285/135;C07D295/14;C07D295/155;C07D295/18;C07D295/20;C07D295/215;C07D307/56;C07D307/68;C07D317/68;C07D333/20;C07D333/38;C07D333/68;C07D401/12;C07D405/06;C07D405/12;C07D409/04;C07D417/04;C07D417/12 主分类号 C07D295/12
代理机构 代理人
主权项
地址