发明名称 |
THE CITRATE SALT OF 5, 8, 14-TRIAZATETRACYCLO(10.3.1.02,11.04.9)-HEXADECA-2.(11),3,5,7,9-PENTAENE AND PHARMACEUTICAL COMPOSITIONS THEREOF |
摘要 |
The present invetion is directed to the citrate salt of 5, 8, 14- triazatetracyclo[10.3.1.02.11.04.9]-hexadeca-2(11),3,5,7,9-pentaene, formula 1, and pharmaceutical compositions thereof. The presetn invention is also directed to the various forms fo the citrate salt, particularly its hydrate and its anhydrous/nearly anyhydrous polmorph. The invention is also directed to processes for preparation of these citrate salt forms. |
申请公布号 |
CA2446988(A1) |
申请公布日期 |
2002.11.21 |
申请号 |
CA20022446988 |
申请日期 |
2002.04.26 |
申请人 |
PFIZER PRODUCTS INC. |
发明人 |
ROSE, PETER ROBERT;JOHNSON, PHILIP JAMES;WINT, LEWIN THEOPHILUS;WILLIAMS, GLENN ROBERT |
分类号 |
C07D487/08;A61K;A61K31/495;A61K31/529;A61P;A61P1/04;A61P3/04;A61P5/14;A61P9/06;A61P9/12;A61P17/00;A61P17/02;A61P25/00;A61P25/04;A61P25/06;A61P25/08;A61P25/10;A61P25/14;A61P25/16;A61P25/18;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P25/30;A61P25/32;A61P25/36;A61P27/00;A61P29/00;A61P31/18;A61P39/02;C07D;C07D221/00;C07D223/00;C07D471/08 |
主分类号 |
C07D487/08 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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