发明名称 |
Process for the synthesis of (3aS)-5,5-dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-c][1,2,4] benzothiadiazine |
摘要 |
Process for the industrial synthesis of (3aS)-5,5-dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo-[2,1-c][1,2,4]benzothiadiazine of formula (I): by enantioselective catalytic hydrogenation of 5,5-dioxo-2,3-dihydro-1H-pyrrolo-[2,1-c][1,2,4]benzothiadiazine. |
申请公布号 |
US2002161222(A1) |
申请公布日期 |
2002.10.31 |
申请号 |
US20020125192 |
申请日期 |
2002.04.18 |
申请人 |
FOUCHER ELSA;THOMINOT GILLES;LECOUVE JEAN-PIERRE;RAMSDEN JAMES ANDREW;COBLEY CHRISTOPHER JAMES |
发明人 |
FOUCHER ELSA;THOMINOT GILLES;LECOUVE JEAN-PIERRE;RAMSDEN JAMES ANDREW;COBLEY CHRISTOPHER JAMES |
分类号 |
C07D513/06;A61K31/549;A61P25/00;A61P25/22;A61P25/24;A61P25/28;C07B61/00;C07D513/04;(IPC1-7):C07D285/34 |
主分类号 |
C07D513/06 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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