发明名称 Inhibitors of neuraminidases
摘要 Disclosed are compounds of the formula:which are useful for inhibiting neuraminidases from disease-causing microorganisms, especially, influenza neuraminidase. Also disclosed are compositions and methods for preventing and treating diseases caused by microorganisms having a neuraminidase, processes for preparing the compounds and synthetic intermediates used in these processes.
申请公布号 US6455571(B1) 申请公布日期 2002.09.24
申请号 US19990421787 申请日期 1999.10.19
申请人 ABBOTT LABORATORIES 发明人 MARING CLARENCE J.;GU YU GUI;CHEN HUI-JU;CHEN YUANWEI;DEGOEY DAVID A.;FLOSI WILLIAM J.;GIRANDA VINCENT L.;GRAMPOVNIK DAVID J.;KATI WARREN M.;KEMPF DALE J.;KENNEDY APRIL;KLEIN LARRY L.;KRUEGER ALLAN C.;LIN ZHEN;MADIGAN DAROLD L.;MCDANIEL KEITH F.;MUCHMORE STEVEN W.;SHAM HING L.;STEWART KENT D.;STOLL VINCENT S.;SUN MINGHUA;TU NOAH P.;WAGENAAR FRANK L.;WANG GARY T.;WANG SHELDON;WIEDEMAN PAUL E.;XU YIBO;YEUNG MING C.;ZHAO CHEN;HANESSIAN STEPHEN;BAYRAKDARIAN MALKEN;LUO XUEHONG
分类号 C07D401/12;A61K31/357;A61K31/40;A61K31/401;A61K31/4025;A61K31/405;A61K31/415;A61K31/4155;A61K31/4178;A61K31/42;A61K31/422;A61K31/425;A61K31/427;A61K31/4439;A61K31/5377;A61K31/66;A61K31/662;A61P31/00;A61P31/12;A61P31/16;A61P43/00;C07D;C07D207/00;C07D207/12;C07D207/16;C07D207/26;C07D207/32;C07D207/327;C07D207/38;C07D207/46;C07D303/16;C07D403/04;C07D403/06;C07D405/04;C07D405/06;C07D407/06;C07D407/12;C07D409/06;C07D413/04;C07D413/06;C07D417/04;C07D417/06;C07D521/00;C07F9/40;C07F9/572;(IPC1-7):A61K31/40;C07D403/02;C07D277/28 主分类号 C07D401/12
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