发明名称 HETEROCYCLIC COMPOUNDS AND THEIR USE AS HISTAMINE H4 LIGANDS.
摘要 A compound of formula (I) wherein: wherein X4 is NR1 or S; _ X1 is CR3; X2 i s NRe or O, provided that X2 is NRe where X1 is N; X3 is N; to treat or preven t disorders ans conditions mediated by the histamine H4 receptor.
申请公布号 CA2440438(A1) 申请公布日期 2002.09.19
申请号 CA20022440438 申请日期 2002.03.08
申请人 ORTHO-MCNEIL PHARMACEUTICAL, INC. 发明人 PIO, BARBARA;SHAH, CHANDRAVADAN R.;LY, KIEV S.;WEI, JIANMEI;KHATUYA, HARIPADA;LOVENBERG, TIMOTHY W.;KREISBERG, JENNIFER D.;EDWARDS, JAMES P.;THURMOND, ROBIN L.;XIAO, WEI;DVORAK, CURT A.;GRICE, CHERYL A.;KARLSSON, LARS;CARRUTHERS, NICHOLAS I.;CHAI, WENYING;SUN, SIQUAN;JABLONOWSKI, JILL A.;KWOK, ANNETTE K.
分类号 C07D307/84;A61K31/496;A61P1/04;A61P7/00;A61P9/06;A61P17/06;A61P19/02;A61P25/28;A61P29/00;A61P37/04;A61P37/06;A61P37/08;A61P43/00;C07D209/42;C07D401/12;C07D403/06;(IPC1-7):C07D209/42;A61K31/404 主分类号 C07D307/84
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