发明名称 PROCESS FOR MAKING SUBSTITUTED 8-ARYLQUINOLINIUM BENZENESULFONATE
摘要 The present invention is directed to a process to synthesize 6-[1-methyl-1-(methylsulfonyl)ethyl]-8-[3(E)-2-[3-methyl-1,2,4-oxadizo l-5-yl]-2-[4-(methylsulfonyl)phenyl]ethenyl]phenyl]quinoline and its benzenesulfonic acid salt.
申请公布号 WO02060897(A2) 申请公布日期 2002.08.08
申请号 WO2001US48385 申请日期 2001.12.14
申请人 MERCK & CO., INC.;DESMOND, RICHARD;CONLON, DAVID, A.;DRAHUS, ANTOINETTE;HO, GUO-JIE;PIPIK, BRENDA;LEBLOND, CARL;VAILAYA, ANANT 发明人 DESMOND, RICHARD;CONLON, DAVID, A.;DRAHUS, ANTOINETTE;HO, GUO-JIE;PIPIK, BRENDA;LEBLOND, CARL;VAILAYA, ANANT
分类号 A61K31/4709;A61P1/00;A61P1/04;A61P7/00;A61P7/12;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P11/08;A61P11/14;A61P13/12;A61P17/00;A61P17/06;A61P19/02;A61P19/10;A61P25/00;A61P25/16;A61P25/24;A61P25/28;A61P27/14;A61P29/00;A61P31/04;A61P35/00;A61P37/06;A61P39/02;C07D413/10 主分类号 A61K31/4709
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