发明名称 BIARYL-OXA(THIA)ZOLE DERIVATIVES AND THEIR USE AS PPARS MODULATORS
摘要 Compounds represented by Formula (I) wherein n is 2, 3, or 4; V is O or S; W is O, S, or SO2 and at least one R5 is a substituted or unsubstituted aryl or a substituted or unsubstituted heteroaryl; are modulators of peroxisome proliferator activated receptors and are useful in the treatment of type II diabetes and of cardiovascular diseases.
申请公布号 WO0116120(A9) 申请公布日期 2002.07.11
申请号 WO2000US23358 申请日期 2000.08.23
申请人 ELI LILLY AND COMPANY;LIGAND PHARMACEUTICALS INCORPORATED;BROOKS, DAWN, A.;RITO, CHRISTOPHER, J.;SHUKER, ANTHONY, J.;DOMINIANNI, SAMUEL, J.;WARSHAWSKY, ALAN, M.;GOSSETT, LYNN, S.;MATTHEWS, DONALD, P.;HAY, DAVID, A.;ARDECKY, ROBERT, J.;MICHELLYS, PIERRE-YVES;TYHONAS, JOHN. S. 发明人 BROOKS, DAWN, A.;RITO, CHRISTOPHER, J.;SHUKER, ANTHONY, J.;DOMINIANNI, SAMUEL, J.;WARSHAWSKY, ALAN, M.;GOSSETT, LYNN, S.;MATTHEWS, DONALD, P.;HAY, DAVID, A.;ARDECKY, ROBERT, J.;MICHELLYS, PIERRE-YVES;TYHONAS, JOHN. S.
分类号 A61K31/421;A61K31/422;A61K31/4439;A61K31/454;A61K31/506;A61K31/5377;A61P3/06;A61P3/10;A61P9/00;A61P25/00;A61P43/00;C07D263/32;C07D277/22;C07D277/24;C07D277/28;C07D277/36;C07D413/10;C07D413/12;(IPC1-7):C07D263/32;A61K31/426;A61K31/427;A61K31/443 主分类号 A61K31/421
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