发明名称 New processes for producing β-alanine derivative.
摘要 The present invention relates to processes for the preparation of beta-alanine derivative shown by following formula (I): wherein R1 is amino protective group, and R2 is acyl group, or a salt thereof, which comprises, subjecting a compound of the formula (II): wherein R1 is the same as defined above, and R3 is protected carboxy, or a salt, to elimination reaction of carboxy protective group, and then to acylation reaction of amino group.
申请公布号 ZA200102781(B) 申请公布日期 2002.07.04
申请号 ZA20010002781 申请日期 2001.04.04
申请人 FUJISAWA PHARMACEUTICAL CO., LTD. 发明人 MITSURU OHKUBO;SATORU KURODA;HIDEKO NAKAMURA;HISASHI TAKASUGI;YOSUKE FUJII;KEIICHI KOGA;EIKI OIKAWA;RYOKI ORII;SHUNSUKE GOTO
分类号 A61K31/455;A61P7/02;C07D211/60 主分类号 A61K31/455
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