发明名称 TREATMENT OF SEXUAL DYSFUNCTION WITH NON PEPTIDE BOMBESIN RECEPTOR ANTAGONISTS
摘要 Bombesin receptor antagonists have been found to be useful in the treatment of sexual dysfunction in both males and females. They may be selective BB1 antagonists or mixed BB1/BB2 antagonists. Combinations are disclosed of bombesin receptor antagonists with a range of other active compounds, for example PDE5 inhibitors, NEP inhibitors and lasofoxifene.
申请公布号 CA2429106(A1) 申请公布日期 2002.05.23
申请号 CA20012429106 申请日期 2001.11.14
申请人 WARNER-LAMBERT COMPANY LLC 发明人 WAYMAN, CHRISTOPHER PETER;VAN DER GRAAF, PIETER HADEWIJN;GONZALEZ, MARIA ISABEL;PINNOCK, ROBERT DENHAM;STOCK, HERMAN THIJS;HIGGINBOTTOM, MICHAEL;NAYLOR, ALISDAIR MARK;PRITCHARD, MARTYN CLIVE
分类号 C07D213/40;A61K31/165;A61K31/17;A61K31/18;A61K31/196;A61K31/395;A61K31/40;A61K31/4015;A61K31/405;A61K31/422;A61K31/433;A61K31/4402;A61K31/4412;A61K31/4439;A61K31/444;A61K31/454;A61K31/4725;A61K31/498;A61K31/506;A61K38/00;A61K45/00;A61K45/06;A61P15/00;A61P15/10;A61P15/12;A61P43/00;C07D209/20;C07D401/12;C07D405/14;C07D409/12;C07D413/12;C07D413/14;C07D417/14;(IPC1-7):A61K31/165 主分类号 C07D213/40
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