发明名称 |
DEHALOGENO COMPOUNDS |
摘要 |
3-(1-Aminocycloalkyl)pyrrolidinyl-substituted-6-dehalogeno(hydrogen- substituted)quinolonecarboxylic acid derivatives having specific substituents as represented by the following general formula (I), salts thereof and hydrates of the same exhibit a broad and potent antibacterial activity on gram- negative and gram-positive bacteria, in particular, resistant bacteria typified by gram-positive cocci including MRSA, PRSP and VRE. Thus, these compounds are usable as drugs.
|
申请公布号 |
CA2429440(A1) |
申请公布日期 |
2002.05.23 |
申请号 |
CA20012429440 |
申请日期 |
2001.11.19 |
申请人 |
DAIICHI PHARMACEUTICAL CO., LTD. |
发明人 |
HAYAKAWA, ISAO;TAKAHASHI, HISASHI;TAKEMURA, MAKOTO;ITOH, MASAO;MIYAUCHI, RIE |
分类号 |
C07D401/04;C07D471/04;C07D498/06;(IPC1-7):C07D498/08;C07D498/04;A61K31/04;A61K38/05;A61K38/06;C07K5/06;C07D491/08;C07K5/10;A61K31/437;A61K31/470;A61K31/538 |
主分类号 |
C07D401/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|