发明名称 2-AMINOPYRIDINE COMPOUNDS AND USE THEREOF AS DRUGS
摘要 <p>2-Aminopyridine compounds of the general formula (I) and salts thereof, exhibiting excellent adenosine receptor (A1, A2a, or A2b receptor) antagonism wherein R1 is cyano, carboxyl, or optionally substituted carbamoyl; R2 is hydrogen, hydroxyl, optionally substituted C¿1-6? alkoxy, an optionally substituted C6-14 aromatic carbocyclic group, or an optionally substituted 5- to 14-membered aromatic heterocyclic group; and R?3 and R4¿ are each independently an optionally substituted C¿6-14? aromatic carbocyclic group, a 5- to 14-membered nonaromatic heterocyclic group, a 5- to 14-membered aromatic heterocyclic group, or the like.</p>
申请公布号 WO2002014282(P1) 申请公布日期 2002.02.21
申请号 JP2001006870 申请日期 2001.08.09
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