发明名称 |
4'-C-ethynyl pyrimidine nucleoside compounds |
摘要 |
The invention provides 4'-C-ethynyl pyrimidine nucleosides (other than 4'-C-ethynylthymidine) represented by formula [I]: wherein B represents a base selected from the group consisting of pyrimidine and derivatives thereof; X represents a hydrogen atom or a hydroxyl group; and R represents a hydrogen atom or a phosphate residue; and a pharmaceutical composition containing any one of the compounds and a pharmaceutically acceptable carrier. Preferably, the composition is used as an anti-HIV agent or a drug for treating AIDS.
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申请公布号 |
US2002022722(A1) |
申请公布日期 |
2002.02.21 |
申请号 |
US20010941845 |
申请日期 |
2001.08.30 |
申请人 |
OHRUI HIROSHI;SHIGETA SHIRO;KODAMA EIICHI;MACHIDA HARUHIKO;KOHGO SATORU;MITSUYA HIROAKI |
发明人 |
OHRUI HIROSHI;SHIGETA SHIRO;KODAMA EIICHI;MACHIDA HARUHIKO;KOHGO SATORU;MITSUYA HIROAKI |
分类号 |
A61P31/18;C07H19/06;C07H19/16;(IPC1-7):C07H19/10 |
主分类号 |
A61P31/18 |
代理机构 |
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地址 |
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