发明名称 6-SUBSTITUTED-7- HETEROQUINOXALINE CARBOXYLIC ACID DERIVATIVES AND ADDITION SALTS THEREOF AND PROCESSES FOR THE PREPARATION OF BOTH
摘要 <p>The invention provides compounds with antagonism against excitatory amino acid receptors, in particular, AMPA receptor having 6-substituted-7-heteroquinoxalinecarboxylic acid derivatives and addition salts thereof as effective ingredients, and processes for the preparation of both. These compounds relate to 6-substituted-7-heteroquinoxalinecarboxylic acid derivatives represented by a general formula (1) &lt;CHEM&gt; (wherein A denotes a single bond or methylene (CH2), Y denotes a nitrogen atom or =CH-, V denotes a single bond or methylene (CH2), T denotes a hydroxyl group, amino group, lower alkoxycarbonyl group, carboxyl group, aldehyde group or the like, Q denotes a halogen atom, lower alkyl group or lower alkoxy group, and R&lt;1&gt; denotes a hydroxyl group, lower alkoxy group or the like), and addition salts thereof.</p>
申请公布号 EP1156047(A1) 申请公布日期 2001.11.21
申请号 EP20000905326 申请日期 2000.02.25
申请人 KYORIN PHARMACEUTICAL CO., LTD. 发明人 TAKANO, YASUO;SHIGA, FUTOSHI;ANRAKU, TSUYOSHI;FUKUCHI, KAZUNORI
分类号 A61P25/00;C07D403/04;A61K31/498;A61P25/28;A61P43/00;C07D403/06;(IPC1-7):C07D403/04 主分类号 A61P25/00
代理机构 代理人
主权项
地址