发明名称 |
BETA-AMINO ACID DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEASES AND TNF-ALPHA |
摘要 |
The present application describes novel &bgr;-amino acid derivatives of formula (I) or pharmaceutically acceptable salt or prodrug forms thereof, wherein A, X, Z, U<a>, X<a>, Y<a>, Z<a>, R<1>, R<2>, R<3>, R<4>, and R<4a> are defined in the present specification, which are useful as metalloprotease and as TNF-&agr; inhibitors.
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申请公布号 |
WO0170734(A2) |
申请公布日期 |
2001.09.27 |
申请号 |
WO2001US08336 |
申请日期 |
2001.03.15 |
申请人 |
DUPONT PHARMACEUTICALS COMPANY |
发明人 |
DUAN, JINGWU;KING, BRYAN, W.;DECICCO, CARL;MADUSKUIE, THOMAS, P., JR.;VOSS, MATTHEW, E. |
分类号 |
A61K31/445;A61K31/4468;A61K31/4545;A61K31/47;A61K31/4709;A61K31/541;A61K31/55;A61P1/02;A61P1/04;A61P1/14;A61P1/16;A61P7/02;A61P7/04;A61P9/00;A61P9/04;A61P11/00;A61P11/06;A61P17/00;A61P17/02;A61P17/06;A61P19/00;A61P19/02;A61P19/04;A61P19/06;A61P19/08;A61P21/00;A61P21/04;A61P25/28;A61P25/32;A61P27/02;A61P27/06;A61P29/00;A61P31/04;A61P31/18;A61P33/02;A61P35/00;A61P35/04;A61P37/00;A61P37/02;A61P39/00;A61P41/00;A61P43/00;C07D211/34;C07D211/58;C07D215/14;C07D401/06;C07D401/12;C07D401/14;C07D405/12;C07D405/14;C07D409/12;C07D413/12;C07D417/12;C07D417/14;C07D451/04;C07D455/02;(IPC1-7):C07D401/12;A61K31/454 |
主分类号 |
A61K31/445 |
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