摘要 |
Antibacterial 3-aminoquinazolin-2,4-diones have formula (I) wherein: R1 and R3 include alkyl, alkenyl, alkynyl, cycloalkyl, aryl, heterocyclic, and heteroaryl; R5, R6, and R8 include H, alkyl, alkoxy, halo, NO2, CN, NH2, alk yl and dialkylamino; R7 includes hydrogen, alkyl, cycloalkyl, heterocyclic, fus ed heterocyclic, aryl and fused aryl; J and K are C or N; and pharmaceutically acceptable salts thereof.
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申请人 |
WARNER-LAMBERT COMPANY |
发明人 |
SHOWALTER, HOWARD DANIEL HOLLIS;WATSON, BRIAN MORGAN;STIER, MICHAEL ANDREW;TRAN, TUAN PHONG;ELLSWORTH, EDMUND LEE;SANCHEZ, JOSEPH PETER;SINGH, RAJESHWAR;BIRD, PAUL;YIP, JUDY;NGUYEN, DAI QUOC |