发明名称 N-SUBSTITUTED ANMINOTETRALINS AS LIGANDS FOR THE NEUROPEPTIDE Y Y5 RECEPTOR USEFUL IN THE TREATMENT OF OBESITY AND OTHER DISORDERS
摘要 Beta-Aminotetralin derivatives of formula which are ligands for the neuropeptide Y Y5 (NPY5) receptor, methods of preparation and pharmaceutical compositions containing a beta-aminotetralin derivative as an active ingredient are described. The beta-aminotetralins are useful in the treatment of disorders and diseases associated with NPY receptor subtype Y5. 22 claims
申请公布号 BG104877(A) 申请公布日期 2001.06.29
申请号 BG20000104877D 申请日期 2000.10.23
申请人 ORTHO-MCNEIL PHARMACEUTICAL INC. 发明人 DAX, SCOTT;LOVENBERG, TIMOTHY W.;MCNALLY, JAMES;REITZ, ALLEN B.;YOUNGMAN, MARK A.
分类号 A61K31/18;A61K31/34;A61K31/341;A61K31/38;A61K31/381;A61K31/415;A61K31/4164;A61K31/44;A61K31/4406;A61K31/4409;A61K31/4418;A61P3/04;A61P3/10;A61P9/00;A61P9/04;A61P9/12;A61P15/00;A61P25/00;A61P25/04;A61P25/06;A61P25/08;A61P25/20;A61P25/22;A61P25/24;A61P25/28;A61P43/00;C07C311/05;C07C311/15;C07C311/18;C07C311/20;C07C311/21;C07C311/22;C07C311/25;C07C311/29;C07C311/37;C07C311/41;C07C317/14;C07D213/16;C07D213/38;C07D233/54;C07D233/64;C07D307/52;C07D333/20;C07D333/34;(IPC1-7):C07C311/15 主分类号 A61K31/18
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