发明名称 Benzoxazinone dopamine D4 receptor antagonists
摘要 Compounds having formulae (I) or (II) wherein R<1> and R<2> are independently hydrogen or C1-C6 alkyl; X is N or CH; and R<3> is phenyl, naphthyl, heteroaryl, substituted phenyl, substituted naphthyl or substituted heteroaryl, wherein each substituent is independently selected from halogen, C1-C6 alkoxy, C1-C6 alkyl, -CN, -CF3, or sulphonamido, and the pharmaceutically acceptable salts, esters, amides, and prodrugs thereof, are antagonists of dopamine D4 receptors.
申请公布号 AU731104(B2) 申请公布日期 2001.03.22
申请号 AU19970030727 申请日期 1997.05.20
申请人 WARNER-LAMBERT COMPANY 发明人 THOMAS BELLIOTTI;LAWRENCE DAVID WISE;DAVID JUERGEN WUSTROW
分类号 A61K31/00;A61K31/535;A61K31/5375;A61K31/5377;A61P25/18;C07D265/36;C07D413/06;C07D413/12;C07D417/12;(IPC1-7):C07D265/36 主分类号 A61K31/00
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