发明名称 3(5)-UREIDO-PYRAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOR AGENTS
摘要 3-ureido-pyrazole derivatives represented by formula (I): where R, R1 and R2 are as described herein, or pharmaceutically acceptable salts thereof; are useful, for example, for the treatment of cancer, cell proliferative disorders, Alzheimer's disease, viral infections, auto-immune diseases or neurodegenerative diseases.
申请公布号 WO0112188(A1) 申请公布日期 2001.02.22
申请号 WO2000US17878 申请日期 2000.08.11
申请人 PHARMACIA & UPJOHN S.P.A.;PHARMACIA & UPJOHN COMPANY;PEVARELLO, PAOLO;ORSINI, PAOLO;TRAQUANDI, GABRIELLA;VARASI, MARIO;FRITZEN, EDWARD, L.;WARPEHOSKI, MARTHA, A.;PIERCE, BETSY, S. 发明人 PEVARELLO, PAOLO;ORSINI, PAOLO;TRAQUANDI, GABRIELLA;VARASI, MARIO;FRITZEN, EDWARD, L.;WARPEHOSKI, MARTHA, A.;PIERCE, BETSY, S.
分类号 C07D231/38;A61K31/415;A61K31/4155;A61K31/4178;A61K31/428;A61K31/4439;A61K31/454;A61K31/4725;A61K31/496;A61K31/498;A61K31/5377;A61P9/10;A61P11/00;A61P13/12;A61P17/06;A61P19/02;A61P35/00;A61P35/02;C07D231/16;C07D231/40;C07D403/12;(IPC1-7):A61K31/415 主分类号 C07D231/38
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