PROCESS FOR THE PREPARATION OF BUTOXYCARBONYLIMINO COMPOUNDS AND INTERMEDIATES THEREFOR
摘要
The present invention relates to a novel process for the preparation of butoxycarbonylimino compounds, in particular (tert-butoxycarbonylimino-pyrazol-1-yl-methyl)-carbamic acid tert-butyl ester, otherwise known as bis-boc-1H-pyrazole-1-carboxamidine, or bis-Boc PC, and novel intermediates.
申请公布号
WO0078723(A1)
申请公布日期
2000.12.28
申请号
WO2000GB02355
申请日期
2000.06.16
申请人
GLAXO GROUP LIMITED;DOWLE, MICHAEL, DENNIS;HOWES, PETER, DAVID;ROBINSON, JOHN, EDWARD;TRIVEDI, NAIMISH