发明名称 |
PROCESS FOR THE PRODUCTION OF TERT-BUTYL (E)-(6-[2- [4-(4-FLUOROPHENYL) -6-ISOPROPYL-2-[ METHYL (METHYLSULFONYL) AMINO] PYRIMIDIN-5-YL] VINYL](4R, 6S)-2,2-DIMETHYL [1,3]DIOXAN-4-YL) ACETATE |
摘要 |
<p>The invention concerns a process for the manufacture of <u>tert</u>-butyl (E)-(6-[2- 4-(4-fluorophenyl) -6-isopropyl-2-[ methyl (met hylsulfonyl) amino] pyrimidin-5-yl] vinyl}-(4R, 6S)-2,2-dimethyl [1,3-dioxan-4-yl) acetate, the novel starting material used in said process and the use of the process in the manufacture of a pharmaceutical.</p> |
申请公布号 |
WO0049014(A1) |
申请公布日期 |
2000.08.24 |
申请号 |
WO2000GB00481 |
申请日期 |
2000.02.15 |
申请人 |
ASTRAZENECA UK LIMITED;SHIONOGI & CO. LTD.;KOIKE, HARUO;KABAKI, MIKIO;TAYLOR, NIGEL, PHILIP;DIORAZIO, LOUIS, JOSEPH |
发明人 |
KOIKE, HARUO;KABAKI, MIKIO;TAYLOR, NIGEL, PHILIP;DIORAZIO, LOUIS, JOSEPH |
分类号 |
A61K31/505;A61P3/06;A61P9/00;A61P9/10;C07D239/00;C07D239/42;C07D319/06;C07D319/08;C07D405/06;C07F9/53;C07F9/6512;(IPC1-7):C07D405/06 |
主分类号 |
A61K31/505 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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