发明名称 |
Method for preparing an aza-macrolide with 4'' (r) nh2 |
摘要 |
The subject-matter of the invention is a process for the stereoselective preparation of a compound of general formula I by stereoselective displacement by a nitrogenous nucleophilic compound of the activated alcohol functional group present at this 4'' position in a corresponding derivative of formula II. |
申请公布号 |
AU1987000(A) |
申请公布日期 |
2000.08.01 |
申请号 |
AU20000019870 |
申请日期 |
2000.01.17 |
申请人 |
MERIAL |
发明人 |
PATRICK LEON;FREDERIC LHERMITTE;RONAN GUEVEL;DENIS PAUZE;LAURENT GAREL;GILLES ODDON |
分类号 |
A61K31/70;A61P31/00;C07B61/00;C07H17/08 |
主分类号 |
A61K31/70 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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