发明名称 SUBSTITUTED 2-ARYLIMINO HETEROCYCLES AND COMPOSITIONS CONTAINING THEM, FOR USE AS PROGESTERONE RECEPTOR BINDING AGENTS
摘要 This invention relates to 2-arylimino heterocycles, including 2-arylimino-1, 3- thiazolidines, 2-arylimino-2, 3, 4, 5-tetrahydro-1, 3-thiazines, 2-arylimino - 1, 3-thiazolidin-4-ones, 2-arylimino-1, 3-thiazolidin-5-ones, and 2-arylimin o- 1, 3-oxazolidines, and their use in modulating progesterone receptor mediate d processes, and pharmaceutical compositions for use in such therapies.</SDOAB >
申请公布号 CA2359562(A1) 申请公布日期 2000.07.20
申请号 CA19992359562 申请日期 1999.12.14
申请人 BAYER CORPORATION 发明人 BULLOCK, WILLIAM H.;BRITTELLI, DAVID R.;BRENNAN, CATHERINE R.;CHEN, JINSHAN;DALLY, ROBERT;COLLIBEE, WILLIAM L.;KLUENDER, HAROLD C. E.;WOLANIN, DONALD J.;URBAHNS, KLAUS;BAGI, CEDO M.;JOHNSON, JEFFREY S.;DIXON, BRIAN R.;MASE, CAROL ANN;LIU, PEIYING;REDMAN, ANIKO M.;LATHROP, WILLIAM F.;SCOTT, WILLIAM J.
分类号 C07D233/42;A61K;A61K31/4164;A61K31/421;A61K31/423;A61K31/425;A61K31/426;A61K31/427;A61K31/428;A61K31/429;A61K31/437;A61K31/54;A61K31/55;A61P;A61P5/00;A61P5/24;A61P9/00;A61P9/10;A61P13/00;A61P15/00;A61P15/04;A61P15/08;A61P15/10;A61P15/16;A61P15/18;A61P17/00;A61P19/00;A61P19/10;A61P25/00;A61P25/24;A61P25/28;A61P35/00;A61P41/00;C07D;C07D263/28;C07D263/52;C07D277/18;C07D277/20;C07D277/42;C07D277/54;C07D277/60;C07D279/06;C07D281/02;C07D417/06;C07D417/12;C07D513/04;C07D513/10;(IPC1-7):C07D277/18 主分类号 C07D233/42
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