发明名称 |
METHOD FOR PREPARING (R)- (+) -3 {1- [2-( 4-BENZOYL- 2-(3,4-DIFLUOROPHENYL)MORPHOLIN- 2-YL)ETHYL]- 4-PHENYLPIPERIDIN -4-YL}-1,1- DIMETHYLUREA, ITS SALTS SOLVATES AND/OR HYDRATES |
摘要 |
The invention concerns a method for preparing (R) -(+)- 3{1- [2-(4 -benzoyl- 2- (3,4-difluorophenyl)morpholin -2-yl}ethyl]- 4-phenylpiperidin- 4-yl]-1,1- dimethylurea, its salts solvates and/or hydrates, of formula (I), intermedia te compounds and succinate and fumarate of (R)- (+)-3{1- [2-(4-benzoyl- 2-(3,4- difluorophenyl)morpholin- 2-yl)ethyl]-4- phenylpiperidin-4- yl}-1,1- dimethylurea.
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申请公布号 |
CA2351539(A1) |
申请公布日期 |
2000.07.06 |
申请号 |
CA19992351539 |
申请日期 |
1999.12.14 |
申请人 |
SANOFI-SYNTHELABO |
发明人 |
BURGOS, ALAIN;CABOS, CLAUDE;BONNEFOY, SABRINA;BERNON, FRANCOISE;LUCAS, ERIC;AULOMBARD, ALAIN |
分类号 |
A61K31/5375;A61K31/5377;A61P1/00;A61P9/00;A61P11/00;A61P13/00;A61P25/00;A61P25/04;A61P25/06;A61P29/00;A61P37/00;A61P43/00;C07D265/30;C07D413/06;(IPC1-7):C07D413/06 |
主分类号 |
A61K31/5375 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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