发明名称 |
PYRIDYLTHIO-COMPOUNDS FOR CONTROL OF HELICOBACTER BACTERIUM |
摘要 |
FIELD: organic chemistry. SUBSTANCE: invention describes compounds of the formula (I): <EMI ID=0.1 HE=33 WI=98 TI=CHI> where substituents and symbols have values given in the invention claim and designated for control of Helicobacter bacterium. Indicated new compounds are synthesized either interaction of compound of the formula (II) <EMI ID=0.2 HE=20 WI=24 TI=CHI> with compound of the formula (III) <EMI ID=0.3 HE=33 WI=79 TI=CHI> or interaction of compound of the formula (IV) <EMI ID=0.4 HE=33 WI=61 TI=CHI> with compound of the formula (V) H[[Y-CrH2r]t-[Z-CuH2u]v-R4 (V). Synthesized compounds are oxidized and/or converted to salts and/or obtained salts are converted to free compounds if necessary. EFFECT: improved method of synthesis. 7 cl, 21 tbl, 5 dwg, 43 ex
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申请公布号 |
RU2149872(C1) |
申请公布日期 |
2000.05.27 |
申请号 |
RU19970102557 |
申请日期 |
1995.07.19 |
申请人 |
BYK GUL'DEN LOMBERG KHEMISHE FABRIK GMBKH |
发明人 |
KOL' BERNKHARD;GRUNDLER GERKHARD;ZENN-BIL'FINGER JORG;KHANAUER GUIDO;ZIMON VOL'FGANG-ALEKSANDER;TSIMMERMAN PETER;OPFERKUKH VOL'FGANG |
分类号 |
C07D213/68;A61K31/44;A61K31/4402;A61K31/4418;A61K31/4427;A61K31/443;A61K31/4433;A61K31/47;A61K31/495;A61K31/505;A61K31/506;A61P31/00;A61P31/04;C07D213/00;C07D213/70;C07D213/74;C07D213/80;C07D239/00;C07D307/00;C07D333/00;C07D401/12;C07D401/14;C07D405/14;C07D409/14;C07D417/14;C07D521/00;(IPC1-7):C07D401/12 |
主分类号 |
C07D213/68 |
代理机构 |
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