发明名称 Azole compounds, their production and use
摘要 PCT No. PCT/JP96/00325 Sec. 371 Date Oct. 17, 1996 Sec. 102(e) Date Oct. 17, 1996 PCT Filed Feb. 15, 1996 PCT Pub. No. WO96/25410 PCT Pub. Date Aug. 20, 1996The present invention provides an azole compound represented by the formula (I): wherein Ar is an optionally substituted phenyl group; R1 and R2, the same or different, are a hydrogen atom or a lower alkyl group, or R1 and R2 may combine together to form a lower alkylene group; R3 is a hydrogen atom or an acyl group; X is a nitrogen atom or a methine group; A is Y=Z (Y and Z, the same or different, are a nitrogen atom or a methine group optionally substituted with a lower alkyl group) or an ethylene group optionally substituted with a lower alkyl group; n is an integer from 0 to 2; and Az is an optionally substituted azolyl group, or its salt, which is useful for a prevention and therapy of a fungal infection of a mammal as a antifungal agent.
申请公布号 US6034248(A) 申请公布日期 2000.03.07
申请号 US19960624649 申请日期 1996.10.17
申请人 TAKEDA CHEMICAL INDUSTRIES, LTD. 发明人 ITOH, KATSUMI;OKONOGI, KENJI;TASAKA, AKIHIRO
分类号 C07D403/06;A01N43/653;C07D521/00;(IPC1-7):C07D403/14 主分类号 C07D403/06
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