发明名称 |
2,4-DIAMINOPYRIMIDINE DERIVATIVE |
摘要 |
PURPOSE: The compounds are novel and have important antibacterial properties. The compounds can be used to inhibit or prevent infectious diseases. The compounds have excellent antibacterial activities against multi-resistance gram positive strains and opportunistic infectious pathogens such as Pneumocystis carinii. Also, the compounds represent synergic effects by being administered as a mixture with known antibacterial active materials. CONSTITUTION: The invention relates to the compounds of Formula I, their pharmaceutically useful salts, the uses of the compounds and their salts as therapeutic active materials; drugs based on the materials and producing methods thereof; the uses of the materials as drug and the uses of the materials for producing antibacterial active drugs; and producing methods of the compounds of Formula I and their pharmaceutically allowable salts and intermediates for producing them.
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申请公布号 |
KR20000011053(A) |
申请公布日期 |
2000.02.25 |
申请号 |
KR19987009204 |
申请日期 |
1998.11.14 |
申请人 |
F. HOFFMANN-LA ROCHE AG |
发明人 |
GUERY PHILIPE;STALDER HENRY;BIS PIERRE CHARLES |
分类号 |
A61K31/00;A61K31/505;A61K31/506;A61K31/535;A61K31/5375;A61K31/5377;A61P31/00;A61P31/04;C07D217/06;C07D401/04;C07D401/10;C07D401/14;C07D405/14;C07D409/04;C07D409/14;C07D417/04;C07D417/14;(IPC1-7):C07D401/10 |
主分类号 |
A61K31/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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