PERFLUORINATED ESTERS OF ALKANOYL L-CARNITINE FOR THE PREPARATION OF CATIONIC LIPIDS FOR THE INTRACELLULAR DELIVERY OF PHARMACOLOGICALLY ACTIVE COMPOUNDS
摘要
Perfluorinated esters of alkanoyl L-carnitine of formula (I) are described, said esters are useful as cationic lipids for the intracellular delivery of pharmacologically active compounds.
申请公布号
CA2329659(A1)
申请公布日期
1999.11.11
申请号
CA19992329659
申请日期
1999.05.04
申请人
SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A.
发明人
PUCCI, ANDREA;TINTI, MARIA ORNELLA;PISANO, CLAUDIO;SANTANIELLO, MOSE;CIMA, MARIA GRAZIA;CRITELLI, LUCIA;SCAFETTA, NAZARENO