发明名称 PROCESS FOR THE PREPARATION OF SUFENTANIL DERIVATIVES BY CARBENE ADDITION/AMINOLYSIS OF 4-PIPERIDONE
摘要 A piperidine derivative such as sufentanil is formed in a process which includes dichloro carbene addition to 4-piperidone and subsequent aminolysis to form a 4-amino-4-carbamoyl piperidine (Formula 1).
申请公布号 CA2167912(C) 申请公布日期 1999.11.09
申请号 CA19942167912 申请日期 1994.09.09
申请人 发明人 MATHEW, JACOB
分类号 C07D211/56;C07D211/66;C07D401/06;C07D409/06;C07D491/10;(IPC1-7):C07D409/06 主分类号 C07D211/56
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