发明名称 USE OF TRICYCLIC 1,4-DIHYDRO-1,4-DIOXO-1H-NAPHTALENE DERIVATIVES, RESULTING NOVEL COMPOUNDS AND THERAPEUTICAL USE THEREOF
摘要 The invention concerns the therapeutic use of tricyclic salts and their pharmaceutically acceptable salts having the general formula:in which:A is either a sulfur atom, an oxygen atom, or an R3N radical where R3 is a hydrogen atom, a C1-C5 alkyl radical, or a substituted or unsubstituted aromatic ring, or a substituted or unsubstituted heteroaromatic ring.R1 is either a C1-C5 alkyl radical,or an R4NH radical where R4 is a hydrogen atom, a C1-C5 alkyl radical, or a substituted or unsubstituted aromatic ring, or a substituted or unsubstituted heteroaromatic ring,or an aromatic ring that may or may not be substituted by one or more acceptor or donor groups, or a heteroaromatic ring having one or more heteroatoms, which may or may not be substituted by acceptor or donor groups.R2 is a hydrogen atom, halogen atom, a C1-C5 alkyl radical, an oxygen atom that may or may not be substituted by a C1-C5 alkyl radical, or an NR5R5, radical where R5 and R5, are, independently of each other, a hydrogen atom, an oxygen atom or monovalent C1-C5 organic radicals.
申请公布号 LT4491(B) 申请公布日期 1999.04.26
申请号 LT19980000085 申请日期 1998.06.10
申请人 LABORATOIRE INNOTHERA, SOCIETE ANONYME 发明人 BOUTHERIN-FALSON,ODILE;DESQUAND-BILLIALD,STEPHANIE;FAVROU,ANITA;FINET,MICHEL;TEMBO,OLIVIER;TORREGROSA,JEAN-LUC;YANNIC-ARNOULT,SYLVIE;DOMAGALA-LE-MARQUER,FLORENCE
分类号 A61K31/00;A61K31/415;A61K31/4164;A61K31/4184;A61K31/42;A61K31/421;A61K31/423;A61K31/425;A61K31/428;A61K31/44;A61K31/4427;A61K31/4439;A61P9/00;A61P9/14;A61P25/06;A61P31/00;C07C46/00;C07C50/24;C07C50/32;C07C225/28;C07C225/30;C07D235/02;C07D263/60;C07D277/84;C07D307/00;C07D413/04;C07D417/04;(IPC1-7):C07D235/02;C07C50/00;A61K31/41 主分类号 A61K31/00
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