ARYLALIPHATIC AMINOAMIDES OF PHENOXYACETIC ACID OR SUBSTITUTED PHENOXYACETIC ACIDS HAVING LOCAL-ANESTHETIC AND ANALGETIC ACTIVITY

摘要

FIELD: medicine. SUBSTANCE: present invention describes biologically active compounds, more particularly arylaliphatic aminoazides of general formula I: wherein when R is CH2OC6H5,, then R1 is NC4H8O, and n is 4,5, 6 and 7; R1 is NC5H10,, and n is 4,5,6 and 7; when R is CH2OC6H4CH3-4, then R1 is N(CH3)2,, and n is 4,5,6 and 7; when R is CH2OC6H4CH3-2,, then R1 is NC5H10, and n is 4,5,6 and 7; when R is CH2OC6H4OCH3-2, then R1 is N(CH3)2, and n is 4,5,6 and 7; when R is CH2OC6H4NO2-4, then R1 is N(C2H5)2, and n is 4,5,6,7; when R is CH2OC6H4F-4, then R1 is NC5H10, and n is 4,5,6,7; when R is CH2OC6H4Br-4, then R1 is N(CH3)2,, and n is 4,5,6,7; when R is CH2OC6H4Cl-2, then R1 is NC5H10, and n is 4,5,6 and 7; R1 is N(CH3)2 and n is 4,5,6 and 7; when R is CH2OC6H4Cl-3, then R1 is NC4H8O, and n is 4,5,6 and 7; when R1 is N(CH3)2 and n is 4,5,6 and 7; when R is CH2OC6H4Cl-4, then R1/ is NC4H8O, and n is 4,5,6 and 7; when R1 is NC5H10, and n is 4,5,6,7; when R is CH2OC6H3Cl2-2,4, then R1 is N(CH3)2, and n is 4,5,6 and 7; when R1 is NC5H10, and n is 4,5,6 and 7; when R1 is N(C2H5)2, and n is 4,5,6,7; when R1 is NC4H8O and n is 4,5,6,7; when R is CH2