发明名称 |
CERTAIN DIARYLIMIDAZOLE DERIVATIVES; A NEW CLASS OF NPY SPECIFIC LIGANDS |
摘要 |
Certain diarylimidazoles act as partial agonists or antagonists for NPY receptors, in particular NPY 5 receptors. They are of use, for example in treating loss of appetite. Such compounds bear aryl groups in the 2 position. Many of the compounds are novel.
|
申请公布号 |
CA2294898(A1) |
申请公布日期 |
1999.01.14 |
申请号 |
CA19982294898 |
申请日期 |
1998.07.02 |
申请人 |
PFIZER INC.;NEUROGEN CORPORATION |
发明人 |
THURKAUF, ANDREW;HUTCHISON, ALAN;ELLIOT, RICHARD L.;YUAN, JUN;BLUM, CHARLES A.;HAMMOND, MARLYS |
分类号 |
A61K31/40;A61K31/4164;A61K31/4178;A61K31/4427;A61K31/443;A61K31/4433;A61K31/4439;A61K31/495;A61K31/538;A61K31/5415;A61P3/04;A61P9/00;A61P43/00;C07D233/54;C07D233/64;C07D401/04;C07D403/04;C07D405/04;C07D405/14;C07D409/04;C07D413/04;C07D417/04;(IPC1-7):C07D413/04;A61K31/415;A61K31/44;A61K31/535;A61K31/54 |
主分类号 |
A61K31/40 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|