发明名称 INDOLE DERIVATIVE FUNCTIONING AS 5-HT RECEPTOR ANTAGONIST
摘要 <p>A compound of formula (I) or a salt thereof:wherein:P1 is pyridiyl;P2 is phenyl;A is a bond or a chain of 1 to 5 atoms optionally substituted by C1-6 alkyl;R1 and R2 groups are each independently hydrogen, C1-6alkyl optionally substituted by NR12R13, C2-6alkenyl, C2-6alkynyl, cyano, halogen, CF3, NR12R13, CHO, OCF3, COR14, CH2OR14 or OR14 where R12, R13 and R14 are independently hydrogen or C1-6alkyl;n and m are independently 0, 1 or 2;R3 is hydrogen or C1-6 alkyl;R4 is a group of formula (i):in which:R6 and R7 are independently hydrogen, C1-6 alkyl optionally substituted by one or more fluorine atoms, C1-6alkylthio, C1-6alkoxy or halogen.</p>
申请公布号 CZ9702445(A3) 申请公布日期 1998.09.16
申请号 CZ19970002445 申请日期 1996.01.26
申请人 SMITHKLINE BEECHAM PLC 发明人 GASTER LARAMIE MARY;WYMAN PAUL ADRIAN;MULHOLLAND KEITH RAYMOND;DAVIES DAVID THOMAS;DUCKWORTH DAVID MALCOM;FORBES IAN THOMSON;JONES GRAHAM ELGIN
分类号 A61K31/40;A61K31/44;A61K31/4427;A61K31/443;A61K31/4433;A61K31/475;A61K31/495;A61K31/50;A61K31/505;A61P25/00;A61P25/30;A61P43/00;C07D401/12;C07D401/14;C07D403/12;C07D405/14;C07D409/14;C07D413/12;C07D417/14;(IPC1-7):C07D401/12 主分类号 A61K31/40
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