<p>A stereoselective glycosylation process for preparing beta anomer fluoronucleosides via the SN2 displacement of an anomeric sulfonyloxy group of an alpha anomer enriched fluorocarbohydrate with a nucleobase.</p>
申请公布号
GR3025689(T3)
申请公布日期
1998.03.31
申请号
GR19970403339T
申请日期
1997.12.16
申请人
ELI LILLY AND COMPANY
发明人
CHOU, TA-SEN;POTEET, LAURIE MICHELLE;KJELL, DOUGLAS PATTON;GROSSMAN, CORA SUE;HERTEL, LARRY WAYNE;HOLMES, RICHARD ELMER;JONES, CHARLES DAVID;MABRY, THOMAS EDWARD