发明名称 Synthesis of bisindolylmalimides
摘要 The present invention provides for the reaction of optionally substituted indole-3-acetamides with optionally substituted methyl indole-3-glyoxyl reagent to prepare potent PKC inhibitors. The reaction is very efficient and robust macrocyclization methodology.
申请公布号 AU4157097(A) 申请公布日期 1998.03.06
申请号 AU19970041570 申请日期 1997.08.22
申请人 ELI LILLY AND COMPANY 发明人 MARGARET MARY FAUL;LEONARD L. WINNEROSKI JR.
分类号 C07D403/14;C07D405/14;C07D498/04;C07D498/22 主分类号 C07D403/14
代理机构 代理人
主权项
地址