发明名称 |
Synthesis of bisindolylmalimides |
摘要 |
The present invention provides for the reaction of optionally substituted indole-3-acetamides with optionally substituted methyl indole-3-glyoxyl reagent to prepare potent PKC inhibitors. The reaction is very efficient and robust macrocyclization methodology. |
申请公布号 |
AU4157097(A) |
申请公布日期 |
1998.03.06 |
申请号 |
AU19970041570 |
申请日期 |
1997.08.22 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
MARGARET MARY FAUL;LEONARD L. WINNEROSKI JR. |
分类号 |
C07D403/14;C07D405/14;C07D498/04;C07D498/22 |
主分类号 |
C07D403/14 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|