发明名称 |
5-Substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)-and 3-(piperidin-4-yl)-1H-indoles: new 5-HT1F agonists |
摘要 |
This invention provides novel 5-HT1F agonists of Formula I <IMAGE> I where A-B, R, R1 and X are as defined in the specification, which are useful for the treatment of migraine and associated disorders.
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申请公布号 |
US5708008(A) |
申请公布日期 |
1998.01.13 |
申请号 |
US19960619783 |
申请日期 |
1996.03.20 |
申请人 |
ELI LILLY AND COMPANY |
发明人 |
AUDIA, JAMES EDMUND;DRESSMAN, BRUCE ANTHONY;DROSTE, JAMES JOSEPH;FRITZ, JAMES ERWIN;KALDOR, STEPHEN WARREN;KOCH, DANIEL JAMES;KRUSHINSKI, JR., JOSEPH HERMAN;NISSEN, JEFFREY SCOTT;ROCCO, VINCENT PATRICK;SCHAUS, JOHN MEHNERT;THOMPSON, DENNIS CHARLES |
分类号 |
A61K31/4427;A61K31/443;A61K31/4433;A61K31/445;A61K31/47;A61K31/495;A61K31/535;A61K31/54;A61P25/00;A61P43/00;C07D401/04;C07D401/14;C07D405/14;C07D407/14;C07D409/14;C07D417/14;(IPC1-7):A61K31/445 |
主分类号 |
A61K31/4427 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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