发明名称 5-Substituted-3-(1,2,3,6-tetrahydropyridin-4-yl)-and 3-(piperidin-4-yl)-1H-indoles: new 5-HT1F agonists
摘要 This invention provides novel 5-HT1F agonists of Formula I <IMAGE> I where A-B, R, R1 and X are as defined in the specification, which are useful for the treatment of migraine and associated disorders.
申请公布号 US5708008(A) 申请公布日期 1998.01.13
申请号 US19960619783 申请日期 1996.03.20
申请人 ELI LILLY AND COMPANY 发明人 AUDIA, JAMES EDMUND;DRESSMAN, BRUCE ANTHONY;DROSTE, JAMES JOSEPH;FRITZ, JAMES ERWIN;KALDOR, STEPHEN WARREN;KOCH, DANIEL JAMES;KRUSHINSKI, JR., JOSEPH HERMAN;NISSEN, JEFFREY SCOTT;ROCCO, VINCENT PATRICK;SCHAUS, JOHN MEHNERT;THOMPSON, DENNIS CHARLES
分类号 A61K31/4427;A61K31/443;A61K31/4433;A61K31/445;A61K31/47;A61K31/495;A61K31/535;A61K31/54;A61P25/00;A61P43/00;C07D401/04;C07D401/14;C07D405/14;C07D407/14;C07D409/14;C07D417/14;(IPC1-7):A61K31/445 主分类号 A61K31/4427
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