| 摘要 |
Thioureido-cyclodextrins particularly useful for solubilising antitumoral and antiparasitic agents, and methods for preparing same, are disclosed. The thioureido-cyclodextrins are of formula (I), wherein m is 6, 7 or 8, R<1> is OH or NH-CS-NHR2, with at least one R<1> being NH-CS-NHR2, and R<2> is an alkyl, monosaccharide, oligosaccharide, glycosyl-amino acid or glycopeptide group. Said cyclodextrins are useful for solubilising antitumoral and antiparasitic agents from the taxol family.
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