发明名称 |
6,9-disubstituted benzazepines having alpha -adrenoceptor blocking activity |
摘要 |
PCT No. PCT/US92/06538 Sec. 371 Date Feb. 4, 1994 Sec. 102(e) Date Feb. 4, 1994 PCT Filed Aug. 5, 1992 PCT Pub. No. WO93/03015 PCT Pub. Date Feb. 18, 1993Alpha-adrenergic receptor antagonists having the formula: <IMAGE> which are useful to produce alpha -adrenoceptor antagonism, pharmaceutical compositions including these antagonists, and methods of using these antagonists to produce alpha -adrenoceptor antagonism in mammals.
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申请公布号 |
US5639748(A) |
申请公布日期 |
1997.06.17 |
申请号 |
US19940193075 |
申请日期 |
1994.02.04 |
申请人 |
SMITHKLINE BEECHAM CORPORATION |
发明人 |
DEMARINIS, ROBERT MICHAEL;PFEIFFER, FRANCIS RICHARD |
分类号 |
C07D401/12;C07D403/04;C07D403/06;C07D403/12;C07D405/12;C07D409/12;(IPC1-7):A61K31/55 |
主分类号 |
C07D401/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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