NOVEL FLUORINATED OR HYDROXYLATED PHENYLIMIDAZOLIDINES HAVING ANTI-ANDROGENIC ACTIVITY, METHOD FOR PREPARING SAME, RESULTING INTERMEDIATES, AND PHARMACEUTICAL COMPOSITIONS

摘要

Products of formula (I), wherein R1 and R2 are particularly cyano and trifluoromethyl, R3 is particularly alkyl, alkenyl or alkynyl, optionally substituted by one or more of halogen, cyano or hydroxyl, R4 and R5 either are particularly methyl optionally substituted by fluorine or form particularly a cyclohexyl radical, and X and Y are particularly oxygen, as well as salts and isomers thereof, are disclosed.