发明名称 PROCESSES AND INTERMEDIATES FOR PREPARING 3-(1-PIPERAZINYL)-1,2-BENZISOTHIAZOLE
摘要 The present invention relates to processes for the preparation of 3-(1-piperazinyl)-1,2-benzisothiazole or its pharmaceutically acceptable salt and to novel intermediates used in the process. 3-(1-piperazinyl)-1,2-benzisothiazole is a key intermediate useful for the preparation of ziprasidone.
申请公布号 WO9717336(A1) 申请公布日期 1997.05.15
申请号 WO1996IB01079 申请日期 1996.10.11
申请人 PFIZER INC.;FOX, DARRELL, E.;LAMBERT, JOHN, F.;SINAY, TERRY, G., JR.;WALINSKY, STANLEY, W. 发明人 FOX, DARRELL, E.;LAMBERT, JOHN, F.;SINAY, TERRY, G., JR.;WALINSKY, STANLEY, W.
分类号 C07D295/22;C07C313/16;C07D275/04;C07D295/26;C07D417/04 主分类号 C07D295/22
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