发明名称 d4T polymorphic form I process
摘要 <p>The present invention concerns a novel process using controlled cooling for obtaining d4T polymorphic Form I from a mixture containing one or more of polymorphic Forms I, II and III. Compound d4T has been approved for use in the treatment of AIDS.</p>
申请公布号 EP0749969(A2) 申请公布日期 1996.12.27
申请号 EP19960304030 申请日期 1996.06.04
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 GANDHI, RAJESH BABULAL;BOGARDUS, JOSEPH BALLARD;GAROFALO, PETER MICHAEL;MARR, TIMOTHY RICHARD;PERRONE, ROBERT KEVIN;KAPLAN, MURRAY ARTHUR
分类号 C07D405/04;A61K31/505;A61P31/12;A61P31/18;C07B63/00;C07H19/06;(IPC1-7):C07D405/04;A61K31/70 主分类号 C07D405/04
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