发明名称 |
DIAZEPINONES, THEIR PRODUCTION AND USE |
摘要 |
A compound of general formula (I), wherein A represents a benzene ring, B represents a 6-membered hydrocarbon ring; X represents a lower alkylene, carbonyl or sulfonyl; Y represents a bond, oxygen or N-R1, R1 represents H or an alkyl group, R represents H, an aromatic group, or an alkyl group optionally substituted by an aromatic group; m and n each represents 1-3, or a salt thereof has potent GnRH receptor antagonizing activity.
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申请公布号 |
CA2213510(A1) |
申请公布日期 |
1996.12.05 |
申请号 |
CA19962213510 |
申请日期 |
1996.05.30 |
申请人 |
TAKEDA CHEMICAL INDUSTRIES, LTD. |
发明人 |
OHKAWA, SHIGENORI;KATO, KOICHI;FUJII, NOBUHIRO |
分类号 |
C07D401/14;C07D403/06;(IPC1-7):C07D403/06;C07D403/14;C07D405/14;C07D409/14;C07D413/14;C07D417/14;A61K31/55 |
主分类号 |
C07D401/14 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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