摘要 |
Novel imidazole derivatives as histamine receptor H3 antagonists and/or agonists, preparation thereof and therapeutical uses thereof. Chemical compounds for use as histamine receptor H3 agonists, partial agonists or antagonists, having general formula (Ia) or (Ib), the use thereof for making drugs, and methods for revealing the agonist, partial agonist or antagonist activity of such compounds in vivo, are disclosed. |
申请人 |
INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE M;SOCIETE CIVILE BIOPROJET;SCHWARTZ, JEAN-CHARLES;ARRANG, JEAN-MICHEL;GARBARG, MONIQUE;QUEMENER, AGNES;LECOMTE, JEANNE-MARIE;LIGNEAU, XAVIER;SCHUNACK, WALTER, G.;STARK, HOLGER;PURAND, KATJA;HUELS, ANNETTE;REIDEMEISTER, SYBILLE;ATHMANI, SALAH;GANELLIN, CHARON, ROBIN;PELLOUX-LEON, NADIA;TERTIUX, WASYL;KRAUSE, MICHAEL, C., O.;BASSEM, SADEK |
发明人 |
SCHWARTZ, JEAN-CHARLES;ARRANG, JEAN-MICHEL;GARBARG, MONIQUE;QUEMENER, AGNES;LECOMTE, JEANNE-MARIE;LIGNEAU, XAVIER;SCHUNACK, WALTER, G.;STARK, HOLGER;PURAND, KATJA;HUELS, ANNETTE;REIDEMEISTER, SYBILLE;ATHMANI, SALAH;GANELLIN, CHARON, ROBIN;PELLOUX-LEON, NADIA;TERTIUX, WASYL;KRAUSE, MICHAEL, C., O.;BASSEM, SADEK |