发明名称 IMIDAZOLE DERIVATIVES AS HISTAMINE RECEPTOR H3 (ANT)AGONISTS
摘要 Novel imidazole derivatives as histamine receptor H3 antagonists and/or agonists, preparation thereof and therapeutical uses thereof. Chemical compounds for use as histamine receptor H3 agonists, partial agonists or antagonists, having general formula (Ia) or (Ib), the use thereof for making drugs, and methods for revealing the agonist, partial agonist or antagonist activity of such compounds in vivo, are disclosed.
申请公布号 WO9629315(A3) 申请公布日期 1996.10.24
申请号 WO1996FR00432 申请日期 1996.03.21
申请人 INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE M;SOCIETE CIVILE BIOPROJET;SCHWARTZ, JEAN-CHARLES;ARRANG, JEAN-MICHEL;GARBARG, MONIQUE;QUEMENER, AGNES;LECOMTE, JEANNE-MARIE;LIGNEAU, XAVIER;SCHUNACK, WALTER, G.;STARK, HOLGER;PURAND, KATJA;HUELS, ANNETTE;REIDEMEISTER, SYBILLE;ATHMANI, SALAH;GANELLIN, CHARON, ROBIN;PELLOUX-LEON, NADIA;TERTIUX, WASYL;KRAUSE, MICHAEL, C., O.;BASSEM, SADEK 发明人 SCHWARTZ, JEAN-CHARLES;ARRANG, JEAN-MICHEL;GARBARG, MONIQUE;QUEMENER, AGNES;LECOMTE, JEANNE-MARIE;LIGNEAU, XAVIER;SCHUNACK, WALTER, G.;STARK, HOLGER;PURAND, KATJA;HUELS, ANNETTE;REIDEMEISTER, SYBILLE;ATHMANI, SALAH;GANELLIN, CHARON, ROBIN;PELLOUX-LEON, NADIA;TERTIUX, WASYL;KRAUSE, MICHAEL, C., O.;BASSEM, SADEK
分类号 G01N33/15;A61K31/415;A61K31/47;A61K31/535;A61P1/00;A61P1/04;A61P7/02;A61P9/00;A61P11/00;A61P13/02;A61P15/00;A61P17/00;A61P25/04;A61P25/20;A61P25/24;A61P25/26;A61P25/28;A61P27/02;A61P27/14;A61P27/16;A61P29/00;A61P37/08;A61P43/00;C07D233/54;C07D233/58;C07D233/60;C07D233/64;C07D401/06;C07D405/12;C07D409/12;C07D411/12;C07D413/12;G01N33/567;G01N33/74 主分类号 G01N33/15
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