发明名称 SUBSTITUTED N-CYCLOALKYLMETHYL-1H-PYRAZOLO[3,4-B¦QUINOLIN-4 AMINES AND COMPOSITIONS AND METHODS OF USE THEREOF
摘要 Substituted N-cycloalkylmethyl-1H-pyrazolo¢3,4-b!quinolin-4-ammines, pharmaceutical compositions containing them and methods for a) effecting c-GMP-phosphodiesterase inhibition, b) treating heart failure and/or hypertension, c) reversing or reducing nitrate-induced tolerance, and d) treating angina pectoris, congestive heart disease and myocardial infarction utilizing them.
申请公布号 CA2211317(A1) 申请公布日期 1996.09.19
申请号 CA19962211317 申请日期 1996.03.05
申请人 SANOFI PHARMACEUTICALS, INC. 发明人 DORITY, JOHN A., JR.;KUMAR, VIRENDRA
分类号 A61K31/435;A61P9/00;A61P9/10;A61P9/12;C07D471/04;(IPC1-7):C07D471/04;A61K31/47;A61K31/535 主分类号 A61K31/435
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