发明名称 8-FLUORO-ANTHRACYCLINES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
摘要 8-fluoro-anthracyclines of formula (I) having cis-stereochemistry between the groups 8-F and 9-OH, are described, such compounds present anti-tumor activity. Their preparation and pharmaceutical compositions containing them are also described.
申请公布号 WO9604292(A1) 申请公布日期 1996.02.15
申请号 WO1995EP03061 申请日期 1995.08.01
申请人 A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L.;BRISTOL-MYERS SQUIBB S.P.A.;ANIMATI, FABIO;ARCAMONE, FEDERICO;GIANNINI, GUISEPPE;LOMBARDI, PAOLO;MONTEAGUDO, EDITH 发明人 ANIMATI, FABIO;ARCAMONE, FEDERICO;GIANNINI, GUISEPPE;LOMBARDI, PAOLO;MONTEAGUDO, EDITH
分类号 A61K31/70;A61K31/7028;A61K31/7034;A61K31/704;A61P35/00;C07C46/00;C07C50/36;C07C50/38;C07H15/252;(IPC1-7):C07H15/252 主分类号 A61K31/70
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