发明名称 |
Analogifremgangsmåte for fremstilling av terapeutisk aktive tioalkyltiocefalosporinderivater |
摘要 |
<p>A novel thioalkylthio cephalosporin antibiotic compound of formula I: <CHEM> wherein Acyl is C1 - C12 acyl; Het is optionally substituted monocyclic heteroaromatic group containing one or more hetero atoms; R<1> is a single bond or C1 - C4 alkylene; R2 is a straight or branched C1 - C4 alkylene; X is a sulfur atom or sulfoxide group; and Y is a hydrogen atom or methoxy group, or a pharmaceutically acceptable salt or an amino-, carboxy- and/or hydroxy-protected derivative thereof, a formulation containing the same and a method for treating bacterial infections.</p> |
申请公布号 |
NO178544(B) |
申请公布日期 |
1996.01.08 |
申请号 |
NO19910002821 |
申请日期 |
1991.07.18 |
申请人 |
SHIONOGI & CO LTD |
发明人 |
KUBOTA, TADATOSHI;KUME, MASAHARU |
分类号 |
A61K31/545;A61K31/546;A61P31/00;A61P31/04;C07D249/04;C07D249/08;C07D401/06;C07D501/00;C07D501/04;C07D501/06;C07D501/59;(IPC1-7):C07D501/59 |
主分类号 |
A61K31/545 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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