发明名称 |
COMPOUND WHICH INHIBITS INTERLEUKIN-1 BETA PROTEASE |
摘要 |
Disclosed are compounds, compositions and methods for inhibiting interleukin-1 beta protease activity, the compounds having the formula (I) <CHEM> wherein R1 is an acyl group, as defined herein, A is an amino acid group as defined herein, n is 0-4 and Y is <CHEM> |
申请公布号 |
JPH0725865(A) |
申请公布日期 |
1995.01.27 |
申请号 |
JP19940089532 |
申请日期 |
1994.04.27 |
申请人 |
STERLING WINTHROP INC |
发明人 |
ROORANDO II DOORU;IRENNEGUBU KEE OSHIFUO;SUTANREE JIEI SHIYUMITSUTO;DENTON DABURIYU HOIYAA;TEINA MOOGAN ROSU;PURASADO BUI CHIYATAABUDEYURA;KIYASARIN PII PUROOTEI;MOHAMETSUDO EMU EE AWADO;JIYOSEFU EMU SARUBINO;JIEIMUSU EMU RINKAA;ERITSUKU PII ROTSUJI;JIYASUBAA SHIN;MAAKU EE EITAA |
分类号 |
A61K31/165;A61K31/17;A61K31/215;A61K31/235;A61K31/24;A61K31/27;A61K31/34;A61K31/341;A61K31/365;A61K31/38;A61K31/381;A61K31/445;A61K31/47;A61K31/472;A61K31/535;A61K31/5375;A61K31/54;A61K38/00;A61K38/55;A61P1/00;A61P1/16;A61P11/00;A61P19/00;A61P19/02;A61P25/00;A61P29/00;A61P31/04;A61P35/00;A61P37/00;A61P37/06;A61P43/00;C07C229/22;C07C233/51;C07C235/12;C07C237/08;C07C237/22;C07C237/36;C07C271/22;C07C275/16;C07C311/16;C07C311/19;C07D209/42;C07D209/44;C07D211/60;C07D215/48;C07D217/26;C07D223/06;C07D233/54;C07D233/64;C07D233/70;C07D233/88;C07D295/08;C07D295/092;C07D295/22;C07D295/30;C07D307/33;C07D307/68;C07D333/24;C07D333/36;C07D333/38;C07D453/02;C07K5/04;C07K5/06;C07K5/08;C07K14/81;C12N9/99 |
主分类号 |
A61K31/165 |
代理机构 |
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代理人 |
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地址 |
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