发明名称 |
NOVEL INHIBITORS OF ADENOSINE MONOPHOSPHATE DEAMINASE |
摘要 |
Novel diazepine derivatives which selectively inhibit adenosine monophosphate deaminase and methods of preparing these compounds are provided. These compounds are useful in treating certain condition in vivo which may be ameliorated by increased local concentrations of adenosine.
|
申请公布号 |
CA2154577(A1) |
申请公布日期 |
1994.08.18 |
申请号 |
CA19942154577 |
申请日期 |
1994.02.03 |
申请人 |
GENSIA, INC. |
发明人 |
ERION, MMARK DAVID;BOOKSER, BRETT CARDER;KASIBHATLA, SRINIVAS RAO;GRUBER, HARRY EDWARD |
分类号 |
A61K31/00;A61K31/55;A61P7/02;A61P9/00;A61P9/10;A61P25/04;A61P29/00;A61P43/00;C07D487/04;(IPC1-7):C07D487/04;C07F9/656;A61K31/675 |
主分类号 |
A61K31/00 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|