发明名称 AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM
摘要 The invention relates to new amino acid derivatives of general formula T - Z - NR1 - (R2CR3) - CO - Y - (CH2)n - R (I) wherein R, R1 to R3, T, Z, Y and N are defined as in claim 1, the diastereomers, enantiomers and salts thereof, particularly the physiologically acceptable salts thereof with inorganic or organic acids or bases, which constitute valuable NPY-antagonistic substances, pharmaceutical compositions containing these compounds, the use thereof and processes for preparing them.
申请公布号 CA2153582(A1) 申请公布日期 1994.08.04
申请号 CA19942153582 申请日期 1994.01.18
申请人 DR. KARL THOMAE GESELLSCHAFT MIT BESCHR NKTER HAFTUNG 发明人 RUDOLF, KLAUS;EBERLEIN, WOLFGANG;ENGEL, WOLFHARD;MIHM, GERHARD;DOODS, HENRI;WIELAND, HEIKE-ANDREA;WILLIM, KLAUS-DIETER;KRAUSE, JUERGEN;DOLLINGER, HORST;ESSER, FRANZ;SCHNORRENBERG, GERD;ENTZEROTH, MICHAEL;WIENEN, WOLFGANG
分类号 A61K31/155;A61K31/165;A61K31/195;A61K31/198;A61K31/38;A61K31/381;A61K31/40;A61K31/403;A61K31/404;A61K31/41;A61K31/415;A61K31/4184;A61K31/4245;A61K31/44;A61K31/4409;A61K31/4418;A61K31/4427;A61K31/445;A61K31/4465;A61K31/4468;A61K31/454;A61K31/47;A61K38/00;A61P9/12;A61P43/00;C07C237/22;C07C237/42;C07C255/60;C07C257/12;C07C257/14;C07C257/18;C07C259/10;C07C259/18;C07C261/04;C07C275/40;C07C279/10;C07C279/12;C07C279/14;C07C279/18;C07C279/36;C07C307/02;C07C307/10;C07C311/08;C07C311/15;C07C311/19;C07C311/39;C07C311/42;C07D209/14;C07D209/16;C07D209/42;C07D209/44;C07D211/28;C07D213/38;C07D213/55;C07D215/12;C07D215/38;C07D223/20;C07D233/24;C07D233/48;C07D233/54;C07D233/64;C07D233/66;C07D233/72;C07D233/88;C07D235/06;C07D235/08;C07D249/08;C07D249/10;C07D249/12;C07D249/14;C07D271/06;C07D271/07;C07D295/15;C07D333/20;C07D333/36;C07D401/12;C07D471/04;C07K5/072;(IPC1-7):C07C279/12;C07D215/14;A61K31/16;C07D333/24;A61K31/33;C07C311/47 主分类号 A61K31/155
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