发明名称 |
AMINO ACID DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS AND PROCESSES FOR PREPARING THEM |
摘要 |
The invention relates to new amino acid derivatives of general formula T - Z - NR1 - (R2CR3) - CO - Y - (CH2)n - R (I) wherein R, R1 to R3, T, Z, Y and N are defined as in claim 1, the diastereomers, enantiomers and salts thereof, particularly the physiologically acceptable salts thereof with inorganic or organic acids or bases, which constitute valuable NPY-antagonistic substances, pharmaceutical compositions containing these compounds, the use thereof and processes for preparing them.
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申请公布号 |
CA2153582(A1) |
申请公布日期 |
1994.08.04 |
申请号 |
CA19942153582 |
申请日期 |
1994.01.18 |
申请人 |
DR. KARL THOMAE GESELLSCHAFT MIT BESCHR NKTER HAFTUNG |
发明人 |
RUDOLF, KLAUS;EBERLEIN, WOLFGANG;ENGEL, WOLFHARD;MIHM, GERHARD;DOODS, HENRI;WIELAND, HEIKE-ANDREA;WILLIM, KLAUS-DIETER;KRAUSE, JUERGEN;DOLLINGER, HORST;ESSER, FRANZ;SCHNORRENBERG, GERD;ENTZEROTH, MICHAEL;WIENEN, WOLFGANG |
分类号 |
A61K31/155;A61K31/165;A61K31/195;A61K31/198;A61K31/38;A61K31/381;A61K31/40;A61K31/403;A61K31/404;A61K31/41;A61K31/415;A61K31/4184;A61K31/4245;A61K31/44;A61K31/4409;A61K31/4418;A61K31/4427;A61K31/445;A61K31/4465;A61K31/4468;A61K31/454;A61K31/47;A61K38/00;A61P9/12;A61P43/00;C07C237/22;C07C237/42;C07C255/60;C07C257/12;C07C257/14;C07C257/18;C07C259/10;C07C259/18;C07C261/04;C07C275/40;C07C279/10;C07C279/12;C07C279/14;C07C279/18;C07C279/36;C07C307/02;C07C307/10;C07C311/08;C07C311/15;C07C311/19;C07C311/39;C07C311/42;C07D209/14;C07D209/16;C07D209/42;C07D209/44;C07D211/28;C07D213/38;C07D213/55;C07D215/12;C07D215/38;C07D223/20;C07D233/24;C07D233/48;C07D233/54;C07D233/64;C07D233/66;C07D233/72;C07D233/88;C07D235/06;C07D235/08;C07D249/08;C07D249/10;C07D249/12;C07D249/14;C07D271/06;C07D271/07;C07D295/15;C07D333/20;C07D333/36;C07D401/12;C07D471/04;C07K5/072;(IPC1-7):C07C279/12;C07D215/14;A61K31/16;C07D333/24;A61K31/33;C07C311/47 |
主分类号 |
A61K31/155 |
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