发明名称 Cyano piperazinyl quinoxaline deriv. prepn.
摘要 2-Cyano 3-piperazinyl qunoxalines of formula (I), which are selective antagonists of 5HT3 receptors and useful for treatment of nausea, vomiting, gastric complaints, anxiety states and pyschotic reactions, are made by replacing halogen in 2-cyano 3-halo quinoxalines with a substituted piperazinyl gp.
申请公布号 ES2042395(A1) 申请公布日期 1993.12.01
申请号 ES19920000430 申请日期 1992.02.27
申请人 PROMOTORA CATALANA DE INVERSIO 发明人 CALDERO GES JOSE MARIA;MONGE VEGA ANTONIO;DEL RIO ZAMBRANA JOAQUIN;PALOP CUBILLO JUAN ANTONIO;LASHERAS ALDAZ BERTA;DEL CASTILLO NIETO JUAN CARLOS;ROCA ACIN JUAN;BOSCH ROVIRA ANNA
分类号 A61K31/495;C07D403/04;(IPC1-7):C07D403/04 主分类号 A61K31/495
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