发明名称 Benzo b thiophen-5-yl derivative and process for producing the same.
摘要 <p>This invention relates to a process for producing a compound represented by formula (6a) or (6b): <CHEM> or <CHEM> wherein R<2> represents a hydrogen atom or a hydroxyl-protecting group and R<4> and R<5>, which may be the same or different, represent lower alkyl groups, using a compound represented by formula (2a) or (2b) obtained by preferential crystallization: <CHEM> or <CHEM> and also to a compound represented by the following formula (7) which is an intermediate useful for producing the compound of formula (6a) or (6b): <CHEM> wherein R<1> represents a group represented by formula (8): <CHEM> wherein R<2> is as defined above and R<3> represents a hydrogen atom or a hydroxyl-protecting group, a group represented by the formula (9): <CHEM> or a group represented by formula (10): <CHEM> wherein R<2> is as defined abovef</p>
申请公布号 EP0565965(A2) 申请公布日期 1993.10.20
申请号 EP19930105441 申请日期 1993.04.01
申请人 TOYAMA CHEMICAL CO., LTD. 发明人 NAKANO, JOJI;TAYA, NOBUHISA;CHAKI, HISAAKI;YAMAFUJI, TETSUO;MOMONOI, KAISHU
分类号 C07D409/04;A61K31/38;A61K31/381;A61P25/28;C07D333/54;C07D333/56;C07D333/58;C07D333/60;C07F7/18;(IPC1-7):C07D333/56 主分类号 C07D409/04
代理机构 代理人
主权项
地址