发明名称 |
Benzo b thiophen-5-yl derivative and process for producing the same. |
摘要 |
<p>This invention relates to a process for producing a compound represented by formula (6a) or (6b): <CHEM> or <CHEM> wherein R<2> represents a hydrogen atom or a hydroxyl-protecting group and R<4> and R<5>, which may be the same or different, represent lower alkyl groups, using a compound represented by formula (2a) or (2b) obtained by preferential crystallization: <CHEM> or <CHEM> and also to a compound represented by the following formula (7) which is an intermediate useful for producing the compound of formula (6a) or (6b): <CHEM> wherein R<1> represents a group represented by formula (8): <CHEM> wherein R<2> is as defined above and R<3> represents a hydrogen atom or a hydroxyl-protecting group, a group represented by the formula (9): <CHEM> or a group represented by formula (10): <CHEM> wherein R<2> is as defined abovef</p> |
申请公布号 |
EP0565965(A2) |
申请公布日期 |
1993.10.20 |
申请号 |
EP19930105441 |
申请日期 |
1993.04.01 |
申请人 |
TOYAMA CHEMICAL CO., LTD. |
发明人 |
NAKANO, JOJI;TAYA, NOBUHISA;CHAKI, HISAAKI;YAMAFUJI, TETSUO;MOMONOI, KAISHU |
分类号 |
C07D409/04;A61K31/38;A61K31/381;A61P25/28;C07D333/54;C07D333/56;C07D333/58;C07D333/60;C07F7/18;(IPC1-7):C07D333/56 |
主分类号 |
C07D409/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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